Protein Details: Voltage gated sodium channel protein type 10 subunit alpha

Protein ID

ICDB_Pro_0330

Protein Name

Voltage gated sodium channel protein type 10 subunit alpha

Gene Name

Scn10a; Sns

Organism

Onychomys torridus (Southern grasshopper mouse)

Length

1959 amino acids

AlphaFoldDB

AF-P0DMA5-F1-model_v4.pdb

Function

Tetrodotoxin-resistant channel that mediates the voltage-dependent sodium ion permeability of excitable membranes. Assuming opened or closed conformations in response to the voltage difference across the membrane; the protein forms a sodium-selective channel through which sodium ions may pass in accordance with their electrochemical gradient. Plays a role in neuropathic pain mechanisms.

Sequence

MEFPIGSVGTTNFRRFTPESLAEIEKQIAAHGAAKKARAKHGERKGQDEKPRPQLDLKACNQLPRFYGELPAELVGEPLEDLDPFYSTHRTFMVLNKGRTISRFSATWALWLFSPFNLIRRTAIKVSVHAWFSIFITITILFNCVCMTQNDLPEKIEYAFTVIYTFEALIKILARGFCLNEFTYLRDPWNWLDFSVITLAYVGAAIDLRGISGLRTFRVLRALKTVSVIPGLKVIVGALIHSVRKLADVTILTVFCLSVFALVGLQLFKGNLKNKCIKRSTDPHNAYNFSSQMADNFYIKNGTTEPLLCGNGSDAGHCPSGYICLKTSDNPDFNYTSFDSFAWAFLSLFRLMTQDSWERLYQQTLRASGKMYMVFFVLVIFLGSFYLVNLILAVVTMAYEEQNQATIAEIEAKEKKFQEALEVLQKEQEVLAALGIDTTSLHSHNGSPLAPKNANERKHRIKSRVSEGSTDDNRSPQSDPYNQRRMSFLGLSSGRRRASHSSVFHFRAPSQDVSFPDGITDDGVFHGDHESHRSSLLLARGAGQAGPLPRSPLASSPNPGPGHREEGQLTAPTGELTTGAPEDLALEAAGQKKNFLSAEYLNEPFRAQRAMSVVSIMTSVIEELEESKLRCPPCLINLAQKYLIWECCPKWMKFKMVLFELVTDPFAELTITLCIVVNTIFMAMEHYPMTDAFDAMLQAGNIVFTVFFTMEMAFKIIAFDPYYYFQKKWNVFDCVIVTVSLLELSIAKKGSLSVLRTFRLLRVFKLAKSWPTLNTLIKIIGNSVGALGNLTFILAIIVFIFALVGKQLLGEDYGCRKDGTALWNEGQLRWHMCDFFHSFLVIFRILCGEWIENMWVCMQVSEKSICLILFLTVMVLGNLVVLNLFIALLLNSFSADNLTAPEDDGEVNNLQVALARTQAFGQRASQAISSYFSSHCRLRWPKVGSQLGVKPSLTSSKAEHHITADAVNTAVGTSAKPALSGPKEDPRDFITDANVWVSVPIAEGESDLDELEEDIEQNSQSSWREESPKGQQDQLWQIQRCEDHQVPNSPGSGMSSEDLASYLGERWKSEATPQVPAEGVDDTSSSEGSTVDCPDPEEILKKIPELADDLEEPDDCFTEGCTRHCPCCKVSTSKFPWTTGWQVRKTCYRIVEHSWFESFIIFMILLSSGALAFEDNYLEQKPRVKSMLEYTDRVFTFIFVFEMLLKWVAYGFKKYFTNAWCWLDFLIVNISLTSLIAKILDYSDVASLKALRTLRALRPLRALSRFEGMRVVVDALVGAIPSIMNVLLVCLIFWLIFSIMGVNLFAGKFSRCIDTSNNPFSVVNSTIVNNKSECRNQNHTGHFFWVNVKVNFDNVAMGYLALLQVATFKGWMDIMYAAVDSREINSQPQWEDNLYMYLYFVVFIIFGGFFTLNLFVGVIIDNFNQQKKKLGGQDIFMTEEQKKYYNAMKKLGSKKPQKPIPRPLNKYQGFVFDIVTRQAFDIIIMVLICLNMITMMVETDGQSEEKTKILGRINQFFVAVFTGECVMKMFALRQYYFTNGWNVFDFIVVILSIGSLVFSAILKSLESYFSPTLFRVIRLARIGRILRLIRAAKGIRTLLFALMMSLPALFNIGLLLFLVMFIYSIFGMASFANVVEEAGIDDMFNFQTFGNSMLCLFQITTSAGWDGLLSPILNTGPPYCDPNLSNNNTSKGNCGSPTVGIVFFTTYIIISFLIVVNMYIAVILENFNVATEESTEPLSEDDFDMFYETWEKFDPEATQFIAFSALSDFADTLSGPLRIPKPNQNILIQMDLPLVPGDKIHCLDILFAFTKNVLGESGELDSLKTNMEEKFMATNLSKASYEPIATTLRWKQEDISATVIQKAYRSYVLQRSLTLSNPLRVPRAEDDDAPLPGEGYVTFMANDSGRLPDKSETTSATSFPPSYDSVTRGLSDRVNISTSNSMHNEDEVTSKEGDSPGPQ

PDB Structures

Ligand Binding

1. DICL_CP

2. DICL_Pep

Binding Site

Disease

neuropathic pain

Location

Plays a role in neuropathic pain mechanisms

DOI ID

10.1126/science.1236451

RefSeq

Feature